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DSpaceUnipr
DSpaceUnipr is the institutional repository of the University of Parma. Its aim is to give visibility to the University's scholarly content and learning material.
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Tesi di dottorato e di master
Scienze del farmaco, delle biolomolecole e dei prodotti per la salute. Tesi di dottorato
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Issue Date
Title
Author(s)
Type
5-Mar-2018
Application of enhanced sampling methods in drug design
Lodola, Alessio
;
Callegari, Donatella
Doctoral thesis
Mar-2020
Inhibition of FGFR and EGFR signalling by ligand traps and kinase inhibitors for anti-cancer drug discovery
Mor, Marco
;
Marseglia, Giuseppe
Doctoral thesis
Mar-2020
Convergent medicinal chemistry approaches against susceptible and resistant mycobacterial infections
Costantino, Gabriele
;
Girardini, Miriam
Doctoral thesis
Mar-2019
An integrated approach for physico-chemical profiling in drug discovery
Vacondio, Federica
;
Ferlenghi, Francesca
Doctoral thesis
Mar-2019
Design, synthesis and optimization of inhibitors of enzymes involved in the sulfur assimilation pathway in Gram negative Bacteria
Costantino, Gabriele
;
Pinto de Magalhães, Joana Rita
Doctoral thesis
Mar-2019
Synthesis of irreversible tyrosine kinase inhibitors and ligand traps as diverse approaches in the antiproliferative therapy
Rivara, Silvia
;
Bozza, Nicole
Doctoral thesis
Apr-2021
Synthesis of new potential inhibitors for the enzyme N-Acylethanolamine Acid Amidase and investigation of substrate specificity
Piomelli, Daniele
;
Ghidini, Andrea
Doctoral thesis
2022
Novel Adjuvant Strategies to overcome Antimicrobial Resistance
Costantino, Gabriele
;
Pavone, Marialaura
Doctoral thesis
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Author
1
Bozza, Nicole
1
Callegari, Donatella
1
Ferlenghi, Francesca
1
Ghidini, Andrea
1
Girardini, Miriam
1
Marseglia, Giuseppe
1
Pavone, Marialaura
1
Pinto de Magalhães, Joana Rita
Subject
1
acquired resistance
1
cancer
1
covalent drugs
1
cysteine
1
dissociation constants
1
drug design
1
drug discovery
1
Efflux Pumps Inhibtors
1
EGFR
1
enhanced sampling
.
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Date issued
3
2019
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2020
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2018
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2021
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2022